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Wayne Shared "Pharmacology Bliss 5/31/24" - 51 Picmonics

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Pharmacology Bliss 5/31/24

Types of Seizures
Tonic-Clonic
Tonic
Clonic
Absence (Petit Mal)
Myoclonic
Atonic
Partial (Focal) Seizure
Focal Aware (Formerly Called Simple Partial)
Focal Impaired Awareness (Formerly Called Complex Partial)
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3 mins
Carbamazepine
Indications
First-line Seizure Medication
First Line for Trigeminal Neuralgia
Mechanism of Action
Stabilizes Inactive State of Na+ Channels
Side Effects
Stevens-Johnson Syndrome
Induce Cytochrome P450
Teratogen
Hepatotoxicity
Blood Dyscrasias
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2 mins
Phenytoin
Indications
Status Epilepticus
Tonic-Clonic Seizures
Mechanism of Action
Blocks Na+ Channel Activation
Inhibition of Glutamate Release
Class IB Antiarrhythmic
Side Effects
Teratogenic
Macrocytic Megaloblastic Anemia
Induce Cytochrome P450
Drug-induced Lupus
Neuropathy
Hirsutism
Gingival Hyperplasia
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1 min
Barbiturates
Barb- Drug Names
Indications
Seizure Treatment
Anesthesia Induction
Mechanism of Action
Increased Duration of Cl- Channel Opening
Decrease Neuron Firing
Side Effects
Sedation
Cardiovascular and Respiratory Depression
CNS Depression
P450 inducer
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2 mins
Benzodiazepines Overview
Indications
First Line for Status Epilepticus
Anesthesia Induction
Anxiety
Eclampsia
Detoxification
Mechanism of Action
'-zepam' and '-zolam' Suffix
Increase Frequency of Cl- Channel Opening
Side Effects
Decrease REM Sleep
CNS Depression
Dependence
Antidote
Flumazenil for Overdose
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2 mins
Lamotrigine
Indications
Seizure Treatment
Bipolar Disorder
Mechanism of Action
Blocks Voltage-Gated Na+ Channels
Side Effect
Stevens-Johnson Syndrome
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1 min
Topiramate
Indications
Seizure Treatment
Migraine Prophylaxis
Mechanism of Action
Increase GABA Action
Blocks Voltage-Gated Na+ Channels
Side Effects
Kidney Stones
Weight Loss
Sedation
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1 min
Adjunct Agents for Partial Seizures (Part 1)
Clorazepate (tranxeme)
Felbamate (Felbatol)
Blocks glycine coactivation
Gabapentin (Neurontin)
Increase release of GABA
Tigabine (Gabatril)
Block GABA reuptake
Levetiracetam (Keppra)
Block neuronal transmission
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1 min
Ethosuximide
Indications
First Line Absence Seizure Treatment
Mechanism of Action
Blocks Thalamic T-Type Ca2+ Channels
Side Effects
Stevens-Johnson Syndrome
Fatigue
Diarrhea
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32 secs
First Line Seizure Medications
Generalized seizures
Levetiracetam
Valproic Acid
Lamotrigine
Topiramate
Absence seizures
Ethosuximide
Tonic-Clonic Seizures
Valproic Acid
Focal seizures
Carbamazepine
Phenytoin
Lamotrigine
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2 mins
Valproic Acid
Indications
First Line Tonic-Clonic Seizure Treatment
Bipolar Disorder
Migraine Prophylaxis
Mechanism of Action
Increases GABA Concentration
Blocks Voltage-Gated Na+ Channels
Side Effect
GI Distress
Contraindication
Contraindicated in Pregnancy
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1 min
Valproic Acid (Valproate) Side Effects
V-A-L-P-R-O-A-T-E
Vomiting
Alopecia
Liver Toxicity
Pancreatitis/Pancytopenia
Retain Fat (Weight Gain)
Oedema (Edema)
Appetite Increase
Tremor
Enzyme Inhibitor (P450)
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2 mins
Vigabatrin and Tiagabine
Mechanisms
Increases GABA Concentration
Inhibits GABA Degradation (Vigabatrin)
Inhibits GABA Reuptake (Tiagabine)
Indications
Infantile Spasms
Partial (Focal) Seizure
Side Effects
Permanent Visual Loss (Vigabatrin)
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1 min
Levetiracetam
Mechanism of Action
SV2A Receptor Antagonist
Modulates GABA and Glutamate
Inhibits Voltage-Gated Ca2+ Channels
Indication
Partial (Focal) Seizures
Tonic-Clonic Seizures
Myoclonic Seizures
Side Effects
Psychiatric Symptoms
Lethargy
Headache
Contraindications
Chronic Kidney Disease
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3 mins
Pregabalin (Lyrica)
Mechanism
GABA Analog
Indications
Seizures
Neuropathic Pain
Fibromyalgia
Side Effects
Headache
Dizziness
Ataxia
Somnolence (Fatigue)
Weight Gain
Angioedema
Rhabdomyolysis
Considerations
Dependence
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2 mins
Inhaled Anesthetics
Mechanism of Action
Unknown Mechanism
Inhaled Anesthetic Drugs
HEISMN Drug Name Acronym
Side Effects
Respiratory Depression
Myocardial Depression
Lower Metabolic Demand, Increased Cerebral Blood Flow
Hepatotoxicity (Halothane)
Nephrotoxicity (Methoxyflurane)
Seizure (Enflurane)
Malignant Hyperthermia
Expansion of Trapped Gas
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2 mins
Midazolam
Indications
Sedation
Amnesia
Anxiolytic
Anticonvulsant
Invasive Procedures
MOA
GABA Agonist
Reversal Agent
Flumazenil
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45 secs
IV Anesthetics
Barbiturates
Benzodiazepines
Respiratory Depression
Hypotension
Ketamine
NMDA Receptor Antagonist
Hallucinations
Opioids
Propofol
Potentiates GABA-A
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2 mins
Propofol
Anesthetic
Rapid Onset
Can cause Hypotension
Rapidly Metabolized
Intra- and Extra-hepatic Metabolism
Potentiates GABA-A
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Fentanyl
Mechanism of Action
Opioid Receptor Agonist
High Potency
Indications
Anesthesia Induction
Chronic Pain
Breakthrough Pain
Side Effects
CNS Depression
Respiratory Depression
Constipation
Miosis
Considerations
Addiction
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3 mins

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